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-Structure paper
タイトル | A Unique Approach to Design Potent and Selective Cyclic Adenosine Monophosphate Response Element Binding Protein, Binding Protein (CBP) Inhibitors. |
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ジャーナル・号・ページ | J. Med. Chem., Vol. 60, Page 10151-10171, Year 2017 |
掲載日 | 2017年5月30日 (構造データの登録日) |
![]() | Bronner, S.M. / Murray, J. / Romero, F.A. / Lai, K.W. / Tsui, V. / Cyr, P. / Beresini, M.H. / de Leon Boenig, G. / Chen, Z. / Choo, E.F. ...Bronner, S.M. / Murray, J. / Romero, F.A. / Lai, K.W. / Tsui, V. / Cyr, P. / Beresini, M.H. / de Leon Boenig, G. / Chen, Z. / Choo, E.F. / Clark, K.R. / Crawford, T.D. / Jayaram, H. / Kaufman, S. / Li, R. / Li, Y. / Liao, J. / Liang, X. / Liu, W. / Ly, J. / Maher, J. / Wai, J. / Wang, F. / Zheng, A. / Zhu, X. / Magnuson, S. |
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手法 | X線回折 |
解像度 | 1.3 - 1.44 Å |
構造データ | ![]() PDB-5w0e: ![]() PDB-6axq: ![]() PDB-6ay3: ![]() PDB-6ay5: |
化合物 | ![]() ChemComp-9U4: ![]() ChemComp-HOH: ![]() ChemComp-DMS: ![]() ChemComp-C2Y: ![]() ChemComp-C3J: ![]() ChemComp-EDO: ![]() ChemComp-NA: ![]() ChemComp-C3V: ![]() ChemComp-SO4: ![]() ChemComp-GOL: |
由来 |
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![]() | TRANSCRIPTION REGULATOR/INHIBITOR / CREBBP / Bromodomain / small molecule inhibitor / TRANSCRIPTION REGULATOR-INHIBITOR complex / TRANSFERASE/TRANSFERASE inhibitor / TRANSFERASE-TRANSFERASE inhibitor complex / SBDD |