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-Structure paper
タイトル | Molecular and cellular mechanisms of HIF prolyl hydroxylase inhibitors in clinical trials. |
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ジャーナル・号・ページ | Chem Sci, Vol. 8, Page 7651-7668, Year 2017 |
掲載日 | 2017年8月9日 (構造データの登録日) |
![]() | Yeh, T.L. / Leissing, T.M. / Abboud, M.I. / Thinnes, C.C. / Atasoylu, O. / Holt-Martyn, J.P. / Zhang, D. / Tumber, A. / Lippl, K. / Lohans, C.T. ...Yeh, T.L. / Leissing, T.M. / Abboud, M.I. / Thinnes, C.C. / Atasoylu, O. / Holt-Martyn, J.P. / Zhang, D. / Tumber, A. / Lippl, K. / Lohans, C.T. / Leung, I.K.H. / Morcrette, H. / Clifton, I.J. / Claridge, T.D.W. / Kawamura, A. / Flashman, E. / Lu, X. / Ratcliffe, P.J. / Chowdhury, R. / Pugh, C.W. / Schofield, C.J. |
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手法 | X線回折 |
解像度 | 1.99 - 2.45 Å |
構造データ | ![]() PDB-5op6: ![]() PDB-5op8: ![]() PDB-5opc: ![]() PDB-5ox5: ![]() PDB-5ox6: |
化合物 | ![]() ChemComp-ZN: ![]() ChemComp-SO4: ![]() ChemComp-A0W: ![]() ChemComp-GOL: ![]() ChemComp-HOH: ![]() ChemComp-A1H: ![]() ChemComp-A1Z: ![]() ChemComp-MN: ![]() ChemComp-B2E: ![]() ChemComp-BCT: |
由来 |
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![]() | OXIDOREDUCTASE / ON-HEME / DIOXYGENASE / OXYGENASE / DNA-BINDING / METAL-BINDING / TRANSCRIPTION / HELIX-LOOP-HELIX-BETA / DSBH / FACIAL TRIAD / ASPARAGINYL/ASPARTYL HYDROXYLASE / EPIGENETIC REGULATION / SIGNALING / ARD / BETA-HYDROXYLATION / ACTIVATOR-INHIBITOR / OXIDOREDUCTASE-PEPTIDE COMPLEX / NON-HEME DIOXYGENASE / IRON / 2-OXOGLUTARATE / HYPOXIA-INDUCIBLE FACTOR / HIF / HIF PROLYL HYDROXYLASE DOMAIN 2 / PHD2 / EGLN1 / HYPOXIA / CYTOPLASM / TRANSCRIPTION/EPIGENETIC REGULATION / DEVELOPMENT / CELL STRUCTURE / TRANSCRIPTION ACTIVATOR/INHIBITOR / UBL CONJUGATION / POLYMORPHISM / VITAMIN C / ZINC-FINGER / FAMILIAL ERYTHROCYTOSIS / BREAST CANCER / TRANSCRIPTION COMPLEX |