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-Structure paper
タイトル | Structure-guided development of covalent TAK1 inhibitors. |
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ジャーナル・号・ページ | Bioorg. Med. Chem., Vol. 25, Page 838-846, Year 2017 |
掲載日 | 2015年10月13日 (構造データの登録日) |
![]() | Tan, L. / Gurbani, D. / Weisberg, E.L. / Hunter, J.C. / Li, L. / Jones, D.S. / Ficarro, S.B. / Mowafy, S. / Tam, C.P. / Rao, S. ...Tan, L. / Gurbani, D. / Weisberg, E.L. / Hunter, J.C. / Li, L. / Jones, D.S. / Ficarro, S.B. / Mowafy, S. / Tam, C.P. / Rao, S. / Du, G. / Griffin, J.D. / Sorger, P.K. / Marto, J.A. / Westover, K.D. / Gray, N.S. |
![]() | ![]() ![]() |
手法 | X線回折 |
解像度 | 2.11 - 2.7515 Å |
構造データ | ![]() PDB-5e7r: ![]() PDB-5j7s: ![]() PDB-5j8i: ![]() PDB-5j9l: ![]() PDB-5jh6: ![]() PDB-5jk3: |
化合物 | ![]() ChemComp-5KW: ![]() ChemComp-HOH: ![]() ChemComp-6H3: ![]() ChemComp-6H4: ![]() ChemComp-6HF: ![]() ChemComp-T92: ![]() ChemComp-6L4: |
由来 |
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![]() | TRANSFERASE/TRANSFERASE inhibitor / Mitogen-activated protein kinase kinase kinase 7/TGF-beta-activated kinase 1 and MAP3K7-binding protein 1 / TRANSFERASE-TRANSFERASE inhibitor complex / Mitogen activated protein kinase kinase kinase 7 / TGF-beta activated Kinase 1 and MAP3K7-binding protein 1 chimera / Serine/threonine kinase which act as essential component of the MAP kinase signal transduction pathway |