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-Structure paper
タイトル | Determinants of Activity at Human Toll-like Receptors 7 and 8: Quantitative Structure-Activity Relationship (QSAR) of Diverse Heterocyclic Scaffolds |
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ジャーナル・号・ページ | J. Med. Chem., Vol. 57, Page 7955-7970, Year 2014 |
掲載日 | 2014年5月9日 (構造データの登録日) |
![]() | Yoo, E. / Salunke, D.B. / Sil, D. / Guo, X. / Salyer, A.C.D. / Hermanson, A.R. / Kumar, M. / Malladi, S.S. / Balakrishna, R. / Thompson, W.H. ...Yoo, E. / Salunke, D.B. / Sil, D. / Guo, X. / Salyer, A.C.D. / Hermanson, A.R. / Kumar, M. / Malladi, S.S. / Balakrishna, R. / Thompson, W.H. / Tanji, H. / Ohto, U. / Shimizu, T. / David, S.A. |
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手法 | X線回折 |
解像度 | 2 - 2.1 Å |
構造データ | ![]() PDB-4qbz: ![]() PDB-4qc0: |
化合物 | ![]() ChemComp-NAG: ![]() ChemComp-D80: ![]() ChemComp-HOH: ![]() ChemComp-XG1: |
由来 |
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![]() | RNA BINDING PROTEIN / Leucine rich repeat / Glycosylation / innate immunity / RNA recognition / ssRNA / RNA Binding / Secreted / Structure-based Ligand Design / TLR8 and TLR7 agonist / vaccine adjuvants / RNA Receptor / Antiviral and Antitumor Drug Binding |