タイトル | Selective activation of Epac1 and Epac2 |
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ジャーナル・号・ページ | To be Published |
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掲載日 | 2013年8月28日 (構造データの登録日) |
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著者 | Rehmann, H. |
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リンク | PubMedで検索 |
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手法 | X線回折 |
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解像度 | 2.4 - 3 Å |
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構造データ | PDB-4mgi: Selective activation of Epac1 and Epac2 手法: X-RAY DIFFRACTION / 解像度: 2.8 Å PDB-4mgk: Selective activation of Epac1 and Epac2 手法: X-RAY DIFFRACTION / 解像度: 2.7 Å PDB-4mgy: Selective activation of Epac1 and Epac2 手法: X-RAY DIFFRACTION / 解像度: 2.6 Å PDB-4mgz: Selective activation of Epac1 and Epac2 手法: X-RAY DIFFRACTION / 解像度: 3 Å PDB-4mh0: Selective activation of Epac1 and Epac2 手法: X-RAY DIFFRACTION / 解像度: 2.4 Å |
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化合物 | ChemComp-H07: (2S,4aR,6R,7R,7aR)-6-{6-amino-8-[(4-chlorophenyl)sulfanyl]-9H-purin-9-yl}-7-methoxytetrahydro-4H-furo[3,2-d][1,3,2]dioxaphosphinin-2-ol 2-oxide / 8-pCPT-2′-O-Me-cAMP
ChemComp-HR6: (2S,4aR,6R,7R,7aS)-6-[6-amino-8-(benzylsulfanyl)-9H-purin-9-yl]-2-sulfanyltetrahydro-4H-furo[3,2-d][1,3,2]dioxaphosphinin-7-ol 2-oxide
ChemComp-HR4: (2S,4aR,6R,7R,7aS)-6-{6-amino-8-[(4-fluorobenzyl)sulfanyl]-9H-purin-9-yl}-2-sulfanyltetrahydro-4H-furo[3,2-d][1,3,2]dioxaphosphinin-7-ol 2-oxide
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由来 | - mus musculus (ハツカネズミ)
- homo sapiens (ヒト)
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キーワード | SIGNALING PROTEIN/GTP-BINDING PROTEIN / Guanine Nucleotide Exchange Factor / Nucleotide Binding / SIGNALING PROTEIN-GTP-BINDING PROTEIN complex |
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