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-Structure paper
タイトル | Plant growth regulator daminozide is a selective inhibitor of human KDM2/7 histone demethylases. |
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ジャーナル・号・ページ | J. Med. Chem., Vol. 55, Page 6639-6643, Year 2012 |
掲載日 | 2012年2月8日 (構造データの登録日) |
著者 | Rose, N.R. / Woon, E.C. / Tumber, A. / Walport, L.J. / Chowdhury, R. / Li, X.S. / King, O.N. / Lejeune, C. / Ng, S.S. / Krojer, T. ...Rose, N.R. / Woon, E.C. / Tumber, A. / Walport, L.J. / Chowdhury, R. / Li, X.S. / King, O.N. / Lejeune, C. / Ng, S.S. / Krojer, T. / Chan, M.C. / Rydzik, A.M. / Hopkinson, R.J. / Che, K.H. / Daniel, M. / Strain-Damerell, C. / Gileadi, C. / Kochan, G. / Leung, I.K. / Dunford, J. / Yeoh, K.K. / Ratcliffe, P.J. / Burgess-Brown, N. / von Delft, F. / Muller, S. / Marsden, B. / Brennan, P.E. / McDonough, M.A. / Oppermann, U. / Klose, R.J. / Schofield, C.J. / Kawamura, A. |
リンク | J. Med. Chem. / PubMed:22724510 |
手法 | X線回折 |
解像度 | 2.25 - 2.4 Å |
構造データ | PDB-4ai8: PDB-4ai9: |
化合物 | ChemComp-SO4: ChemComp-GOL: ChemComp-DZA: ChemComp-ZN: ChemComp-HOH: ChemComp-NI: ChemComp-CL: |
由来 |
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キーワード | OXIDOREDUCTASE / DIOXYGENASE / METAL-BINDING / HELIX-LOOP-HELIX-BETA / DSBH / FACIAL TRIAD / TRANSCRIPTION AND EPIGENETIC REGULATION / ANKYRIN REPEAT DOMAIN / BETA-HYDROXYLATION / TRANSCRIPTION ACTIVATOR/INHIBITOR / OXYGENASE / DOUBLE-STRANDED BETA HELIX / EPIGENETIC AND TRANSCRIPTION REGULATION / CHROMATIN REGULATOR / HYDROXYLATION |