タイトル | Structural basis of pharmacological chaperoning for human beta-galactosidase |
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ジャーナル・号・ページ | to be published |
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掲載日 | 2013年7月16日 (構造データの登録日) |
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著者 | Suzuki, H. / Ohto, U. / Higaki, K. / Mena-Barragan, T. / Aguilar-Moncayo, M. / Ortiz Mellet, C. / Nanba, E. / Garcia Fernandez, J.M. / Suzuki, Y. / Shimizu, T. |
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リンク | PubMedで検索 |
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手法 | X線回折 |
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解像度 | 2 - 2.3 Å |
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構造データ | PDB-3wez: Crystal structure of human beta-galactosidase in complex with NOEV 手法: X-RAY DIFFRACTION / 解像度: 2.11 Å PDB-3wf0: Crystal structure of human beta-galactosidase in complex with 6S-NBI-DGJ 手法: X-RAY DIFFRACTION / 解像度: 2.2 Å PDB-3wf1: Crystal structure of human beta-galactosidase in complex with 6S-NBI-GJ 手法: X-RAY DIFFRACTION / 解像度: 2 Å PDB-3wf2: Crystal structure of human beta-galactosidase in complex with NBT-DGJ 手法: X-RAY DIFFRACTION / 解像度: 2.3 Å PDB-3wf3: Crystal structure of human beta-galactosidase mutant I51T in complex with Galactose 手法: X-RAY DIFFRACTION / 解像度: 2.15 Å PDB-3wf4: Crystal structure of human beta-galactosidase mutant I51T in complex with 6S-NBI-DGJ 手法: X-RAY DIFFRACTION / 解像度: 2.3 Å |
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化合物 | ChemComp-6DJ: (3Z,6S,7R,8S,8aS)-3-(butylimino)hexahydro[1,3]thiazolo[3,4-a]pyridine-6,7,8-triol / 6S-NBI-DGJ
ChemComp-6GJ: (3E,5S,6R,7S,8S,8aS)-3-(butylimino)hexahydro[1,3]thiazolo[3,4-a]pyridine-5,6,7,8-tetrol
ChemComp-NDJ: (2R,3S,4R,5S)-N-butyl-3,4,5-trihydroxy-2-(hydroxymethyl)piperidine-1-carbothioamide
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由来 | - homo sapiens (ヒト)
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キーワード | HYDROLASE / GLYCOSYL HYDROLASE / TIM-BARREL DOMAIN |
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