タイトル | Mechanism of AMPA Receptor Activation by Partial Agonists: DISULFIDE TRAPPING OF CLOSED LOBE CONFORMATIONS. |
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ジャーナル・号・ページ | J. Biol. Chem., Vol. 286, Page 35257-35266, Year 2011 |
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掲載日 | 2011年8月2日 (構造データの登録日) |
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著者 | Ahmed, A.H. / Wang, S. / Chuang, H.H. / Oswald, R.E. |
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リンク | J. Biol. Chem. / PubMed:21846932 |
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手法 | X線回折 |
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解像度 | 1.823 - 2.015 Å |
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構造データ | PDB-3t93: Glutamate bound to a double cysteine mutant (A452C/S652C) of the ligand binding domain of GluA2 手法: X-RAY DIFFRACTION / 解像度: 1.907 Å PDB-3t96: Iodowillardiine bound to a double cysteine mutant (A452C/S652C) of the ligand binding domain of GluA2 手法: X-RAY DIFFRACTION / 解像度: 1.872 Å PDB-3t9h: Kainate bound to a double cysteine mutant (A452C/S652C) of the ligand binding domain of GluA2 手法: X-RAY DIFFRACTION / 解像度: 2.015 Å PDB-3t9u: CNQX bound to an oxidized double cysteine mutant (A452C/S652C) of the ligand binding domain of GluA2 手法: X-RAY DIFFRACTION / 解像度: 1.97 Å PDB-3t9v: CNQX bound to a reduced double cysteine mutant (A452C/S652C) of the ligand binding domain of GluA2 手法: X-RAY DIFFRACTION / 解像度: 1.975 Å PDB-3t9x: Glutamate bound to a double cysteine mutant (V484C/E657C) of the ligand binding domain of GluA2 手法: X-RAY DIFFRACTION / 解像度: 1.823 Å |
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化合物 | ChemComp-KAI: 3-(CARBOXYMETHYL)-4-ISOPROPENYLPROLINE / カイニン酸 / 神経伝達物質, アゴニスト*YM
ChemComp-CNI: 7-nitro-2,3-dioxo-2,3-dihydroquinoxaline-6-carbonitrile
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由来 | - rattus norvegicus (ドブネズミ)
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キーワード | TRANSPORT PROTEIN / S1S2 / neurotransmitter receptor |
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