+検索条件
-Structure paper
タイトル | Discovery and Characterization of Non-ATP Site Inhibitors of the Mitogen Activated Protein (MAP) Kinases. |
---|---|
ジャーナル・号・ページ | Acs Chem. Biol., Vol. 6, Page 234-244, Year 2011 |
掲載日 | 2010年6月9日 (構造データの登録日) |
![]() | Comess, K.M. / Sun, C. / Abad-Zapatero, C. / Goedken, E.R. / Gum, R.J. / Borhani, D.W. / Argiriadi, M. / Groebe, D.R. / Jia, Y. / Clampit, J.E. ...Comess, K.M. / Sun, C. / Abad-Zapatero, C. / Goedken, E.R. / Gum, R.J. / Borhani, D.W. / Argiriadi, M. / Groebe, D.R. / Jia, Y. / Clampit, J.E. / Haasch, D.L. / Smith, H.T. / Wang, S. / Song, D. / Coen, M.L. / Cloutier, T.E. / Tang, H. / Cheng, X. / Quinn, C. / Liu, B. / Xin, Z. / Liu, G. / Fry, E.H. / Stoll, V. / Ng, T.I. / Banach, D. / Marcotte, D. / Burns, D.J. / Calderwood, D.J. / Hajduk, P.J. |
![]() | ![]() ![]() |
手法 | X線回折 |
解像度 | 2.51 - 2.7 Å |
構造データ | ![]() PDB-3new: ![]() PDB-3o2m: |
化合物 | ![]() ChemComp-3NE: ![]() ChemComp-46A: ![]() ChemComp-SO4: |
由来 |
|
![]() | TRANSFERASE/TRANSFERASE INHIBITOR / Kinase / Ser/Thr kinase / Intracellular / TRANSFERASE-TRANSFERASE INHIBITOR complex / TRANSFERASE/INHIBITOR / Serine Threonine Protein Kinase / ATP binding / Phosphorylation / Kinase-Inhibitor complex / TRANSFERASE-INHIBITOR complex |