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-Structure paper
タイトル | Family-wide chemical profiling and structural analysis of PARP and tankyrase inhibitors. |
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ジャーナル・号・ページ | Nat. Biotechnol., Vol. 30, Page 283-288, Year 2012 |
掲載日 | 2009年3月20日 (構造データの登録日) |
![]() | Wahlberg, E. / Karlberg, T. / Kouznetsova, E. / Markova, N. / Macchiarulo, A. / Thorsell, A.G. / Pol, E. / Frostell, A. / Ekblad, T. / Oncu, D. ...Wahlberg, E. / Karlberg, T. / Kouznetsova, E. / Markova, N. / Macchiarulo, A. / Thorsell, A.G. / Pol, E. / Frostell, A. / Ekblad, T. / Oncu, D. / Kull, B. / Robertson, G.M. / Pellicciari, R. / Schuler, H. / Weigelt, J. |
![]() | ![]() ![]() |
手法 | X線回折 |
解像度 | 1.5 - 2.8 Å |
構造データ | ![]() PDB-3goy: ![]() PDB-3mhj: ![]() PDB-3mhk: ![]() PDB-3p0n: ![]() PDB-3p0p: ![]() PDB-3p0q: ![]() PDB-3se2: ![]() PDB-3smi: ![]() PDB-3smj: |
化合物 | ![]() ChemComp-3AB: ![]() ChemComp-ZN: ![]() ChemComp-M3F: ![]() ChemComp-SO4: ![]() ChemComp-HOH: ![]() ChemComp-P4L: ![]() ChemComp-GOL: ![]() ChemComp-BPU: ![]() ChemComp-NNF: ![]() ChemComp-NNL: ![]() ChemComp-NA: ![]() ChemComp-LDR: ![]() ChemComp-SCN: ![]() ChemComp-CL: ![]() ChemComp-QDR: ![]() ChemComp-FDR: |
由来 |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / PARP / POLY(ADP-RIBOSE) POLYMERASE / BAL-2 / SGC / STRUCTURAL GENOMICS CONSORTIUM / NAD / TRANSFERASE / Glycosyltransferase / Nucleus / Transcription / Transcription regulation / TRANSFERASE-TRANSFERASE INHIBITOR complex / CATALYTIC FRAGMENT / STRUCTURAL GENOMICS / ADP-RIBOSYLATION / ANK REPEAT / CHROMOSOMAL PROTEIN / GOLGI APPARATUS / MEMBRANE / MRNA TRANSPORT / PHOSPHORYLATION / PROTEIN TRANSPORT / TELOMERE / TRANSLOCATION / TRANSPORT / WNT-SIGNALLING / PROTEIN-LIGAND COMPLEX / diphtheria toxin like fold / NAD+ |