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-Structure paper
タイトル | Design of HIV Protease Inhibitors Based on Inorganic Polyhedral Metallacarboranes |
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ジャーナル・号・ページ | J. Med. Chem., Vol. 52, Page 7132-7141, Year 2009 |
掲載日 | 2009年7月10日 (構造データの登録日) |
著者 | Pokorna, J. / Brynda, J. / Cigler, P. / Fanfrlik, J. / Sieglova, I. / Oberwinkler, H. / Hobza, P. / Kral, V. / Konvalinka, J. |
リンク | J. Med. Chem. / PubMed:19874035 |
手法 | X線回折 |
解像度 | 1.7 Å |
構造データ | PDB-3i8w: |
化合物 | ChemComp-CB5: ChemComp-CL: ChemComp-GOL: ChemComp-HOH: |
由来 |
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キーワード | HYDROLASE/HYDROLASE INHIBITOR / inhibitor / cobalt bis(1 / 2-dicarbollide) / viral resistance / aspartic protease / AIDS / Aspartyl protease / Capsid maturation / Capsid protein / Cell membrane / DNA integration / DNA recombination / DNA-directed DNA polymerase / Endonuclease / Hydrolase / Lipoprotein / Magnesium / Membrane / Metal-binding / Multifunctional enzyme / Myristate / Nuclease / Nucleotidyltransferase / Nucleus / Phosphoprotein / Protease / RNA-binding / RNA-directed DNA polymerase / Transferase / Viral nucleoprotein / Virion / Zinc-finger / HYDROLASE-HYDROLASE INHIBITOR COMPLEX |