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-Structure paper
タイトル | Think twice: understanding the high potency of bis(phenyl)methane inhibitors of thrombin |
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ジャーナル・号・ページ | J. Mol. Biol., Vol. 391, Page 552-564, Year 2009 |
掲載日 | 2007年11月6日 (構造データの登録日) |
![]() | Baum, B. / Muley, L. / Heine, A. / Smolinski, M. / Hangauer, D. / Klebe, G. |
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手法 | X線回折 |
解像度 | 1.58 - 2.25 Å |
構造データ | ![]() PDB-2zc9: ![]() PDB-2zda: ![]() PDB-2zfp: ![]() PDB-2zgx: ![]() PDB-2zo3: ![]() PDB-3dhk: ![]() PDB-3dux: ![]() PDB-3f68: |
化合物 | ![]() ChemComp-NA: ![]() ChemComp-22U: ![]() ChemComp-HOH: ![]() ChemComp-PO4: ![]() ChemComp-32U: ![]() ChemComp-19U: ![]() ChemComp-29U: ![]() ChemComp-33U: ![]() ChemComp-23U: ![]() ChemComp-64U: ![]() ChemComp-91U: |
由来 |
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![]() | BLOOD CLOTTING/HYDROLASE INHIBITOR / Blood Clotting/Serine Protease Inhibitors / Secreted / Sulfation / Acute phase / Blood coagulation / Cleavage on pair of basic residues / Disease mutation / Gamma-carboxyglutamic acid / Glycoprotein / Hydrolase / Kringle / Zymogen / BLOOD CLOTTING-HYDROLASE INHIBITOR COMPLEX / Blood Clotting/Hydrolase Inhibitors / Protease / Serine protease / Hydrolase/Hydrolase Inhibitor / Blood Clotting / Hydrolase Inhibitor / Protease inhibitor / Serine protease inhibitor / Hydrolase-Hydrolase Inhibitor complex |