+検索条件
-Structure paper
タイトル | Differential Binding of Inhibitors to Active and Inactive Cdk2 Provides Insights for Drug Design. |
---|---|
ジャーナル・号・ページ | Chem. Biol., Vol. 13, Page 201-, Year 2006 |
掲載日 | 2005年10月30日 (構造データの登録日) |
![]() | Kontopidis, G. / Mcinnes, C. / Pandalaneni, S.R. / Mcnae, I. / Gibson, D. / Mezna, M. / Thomas, M. / Wood, G. / Wang, S. / Walkinshaw, M.D. / Fischer, P.M. |
![]() | ![]() ![]() |
手法 | X線回折 |
解像度 | 2.1 - 2.9 Å |
構造データ | ![]() PDB-2c5n: ![]() PDB-2c5o: ![]() PDB-2c5v: ![]() PDB-2c5x: ![]() PDB-2c5y: |
化合物 | ![]() ChemComp-CK8: ![]() ChemComp-HOH: ![]() ChemComp-CK2: ![]() ChemComp-CK4: ![]() ChemComp-MTW: |
由来 |
|
![]() | TRANSFERASE / DIFFERENTIAL INHIBITION / CDK2 / ATP-BINDING / CELL CYCLE / CELL DIVISION / POLYMORPHISM / PHOSPHORYLATION / NUCLEOTIDE-BINDING / SERINE/THREONINE-PROTEIN / KINASE / MITOSIS / CYCLIN / COMPLEX (KINASE-CYCLIN) / CYCIN A / DRUG DESIGN / LIGAND EXCHANGE / SERINE/THREONINE-PROTEIN KINASE / COMPLEX (TRANSFERASE-CYCLIN) / TRANSFERASE/INHIBITOR / INHIBITION / ACTIVE / INACTIVE / COMPLEX (TRANSFERASE-INHIBITOR) / TRANSFERASE-INHIBITOR complex |