タイトル Regulatory Roles of the N-Terminal Domain Based on Crystal Structures of Human Pyruvate Dehydrogenase Kinase 2 Containing Physiological and Synthetic Ligands. ジャーナル・号・ページ Biochemistry , Vol. 45, Page 402-, Year 2006掲載日 2005年6月8日 (構造データの登録日) 著者Knoechel, T.R. / Tucker, A.D. / Robinson, C.M. / Phillips, C. / Taylor, W. / Bungay, P.J. / Kasten, S.A. / Roche, T.E. / Brown, D.G. リンク Biochemistry / PubMed:16401071手法 X線回折 解像度 2.2 - 2.5 Å 構造データ PDB-2btz : 構造ビューア crystal structures of human pyruvate dehydrogenase kinase 2 containing physiological and synthetic ligands手法 : X-RAY DIFFRACTION / 解像度 : 2.2 Å
PDB-2bu2 : 構造ビューア crystal structures of human pyruvate dehydrogenase kinase 2 containing physiological and synthetic ligands手法 : X-RAY DIFFRACTION / 解像度 : 2.4 Å
PDB-2bu5 : 構造ビューア crystal structures of human pyruvate dehydrogenase kinase 2 containing physiological and synthetic ligands手法 : X-RAY DIFFRACTION / 解像度 : 2.35 Å
PDB-2bu6 : 構造ビューア crystal structures of human pyruvate dehydrogenase kinase 2 containing physiological and synthetic ligands手法 : X-RAY DIFFRACTION / 解像度 : 2.4 Å
PDB-2bu7 : 構造ビューア crystal structures of human pyruvate dehydrogenase kinase 2 containing physiological and synthetic ligands手法 : X-RAY DIFFRACTION / 解像度 : 2.4 Å
PDB-2bu8 : 構造ビューア crystal structures of human pyruvate dehydrogenase kinase 2 containing physiological and synthetic ligands手法 : X-RAY DIFFRACTION / 解像度 : 2.5 Å
化合物 ChemComp-TF2 : 構造ビューア (N-{4-[(ETHYLANILINO)SULFONYL]-2-METHYLPHENYL}-3,3,3-TRIFLUORO-2-HYDROXY-2-METHYLPROPANAMIDE
ChemComp-TF3 : 構造ビューア N-(2-AMINOETHYL)-2-{3-CHLORO-4-[(4-ISOPROPYLBENZYL)OXY]PHENYL} ACETAMIDE
由来 homo sapiens (ヒト) キーワード TRANSFERASE / GHKL MOTIF REGULATION / PYRUVATE DEHYDROGENASE KINASE 2 / PYRUVATE DEHYDROGENASE KINASE 2 GHKL MOTIF REGULATION