タイトル | Combining mutations in HIV-1 protease to understand mechanisms of resistance. |
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ジャーナル・号・ページ | Proteins, Vol. 48, Page 107-116, Year 2002 |
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掲載日 | 2001年9月25日 (構造データの登録日) |
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著者 | Mahalingam, B. / Boross, P. / Wang, Y.F. / Louis, J.M. / Fischer, C.C. / Tozser, J. / Harrison, R.W. / Weber, I.T. |
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リンク | Proteins / PubMed:12012342 |
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手法 | X線回折 |
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解像度 | 1.2 - 2.2 Å |
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構造データ | PDB-1k1t: Combining Mutations in HIV-1 Protease to Understand Mechanisms of Resistance 手法: X-RAY DIFFRACTION / 解像度: 1.2 Å PDB-1k1u: Combining Mutations in HIV-1 Protease to Understand Mechanisms of Resistance 手法: X-RAY DIFFRACTION / 解像度: 1.55 Å PDB-1k2b: Combining Mutations in HIV-1 Protease to Understand Mechanisms of Resistance 手法: X-RAY DIFFRACTION / 解像度: 1.7 Å PDB-1k2c: Combining Mutations in HIV-1 Protease to Understand Mechanisms of Resistance 手法: X-RAY DIFFRACTION / 解像度: 2.2 Å |
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化合物 | ChemComp-0Q4: N-[(2R)-2-({N~5~-[amino(iminio)methyl]-L-ornithyl-L-valyl}amino)-4-methylpentyl]-L-phenylalanyl-L-alpha-glutamyl-L-alanyl-L-norleucinamide
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由来 | ![](img/tx_virus.gif) human immunodeficiency virus 1 (ヒト免疫不全ウイルス)
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キーワード | HYDROLASE/HYDROLASE INHIBITOR / HIV-1 PROTEASE / HYDROLASE-HYDROLASE INHIBITOR COMPLEX |
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