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-Structure paper
Title | Discovery and binding mode of small molecule inhibitors of the apo form of human TDO2 |
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Journal, issue, pages | To Be Published |
Publish date | Apr 12, 2024 (structure data deposition date) |
![]() | Lotz-Jenne, C. / lange, R. / Cren, S. / Bourquin, G. / Goglia, L. / Kimmerlin, T. / Wicki, M. / Mueller, M. / Artico, N. / Ackerknecht, S. ...Lotz-Jenne, C. / lange, R. / Cren, S. / Bourquin, G. / Goglia, L. / Kimmerlin, T. / Wicki, M. / Mueller, M. / Artico, N. / Ackerknecht, S. / Joesch, C. / Mac Sweeney, A. |
![]() | Search PubMed |
Methods | X-ray diffraction |
Resolution | 2.612 Å |
Structure data | ![]() PDB-9ezj: |
Chemicals | ![]() ChemComp-ZIQ: ![]() PDB-1h8g: ![]() ChemComp-HOH: |
Source |
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![]() | OXIDOREDUCTASE / apo-TDO / heme / inhibitor |