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-Structure paper
Title | Identification and Optimization of Small Molecule Pyrazolopyrimidine TLR7 Agonists for Applications in Immuno-oncology. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 15, Page 189-196, Year 2024 |
Publish date | Mar 28, 2023 (structure data deposition date) |
Authors | He, L. / Zhang, M.Y. / Cox, M. / Zhang, Q. / Donnell, A.F. / Zhang, Y. / Tarby, C. / Gill, P. / Subbaiah, M.A.M. / Ramar, T. ...He, L. / Zhang, M.Y. / Cox, M. / Zhang, Q. / Donnell, A.F. / Zhang, Y. / Tarby, C. / Gill, P. / Subbaiah, M.A.M. / Ramar, T. / Reddy, M. / Puttapaka, V. / Li, Y.X. / Sivaprakasam, P. / Critton, D. / Mulligan, D. / Xie, C. / Ramakrishnan, R. / Nagar, J. / Dudhgaonkar, S. / Murtaza, A. / Oderinde, M.S. / Schieven, G.L. / Mathur, A. / Gavai, A.V. / Vite, G. / Gangwar, S. / Poudel, Y.B. |
External links | Acs Med. Chem. Lett. / PubMed:38352849 |
Methods | X-ray diffraction |
Resolution | 2.437 Å |
Structure data | PDB-8s9h: |
Chemicals | ChemComp-NAG:
ChemComp-ZWV: ChemComp-SO4: ChemComp-HOH: |
Source |
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Keywords | IMMUNE SYSTEM / Toll-like receptor 7 / pattern recognition receptor / agonist |