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Title | Reverse N -Substituted Hydroxamic Acid Derivatives of Fosmidomycin Target a Previously Unknown Subpocket of 1-Deoxy-d-xylulose 5-Phosphate Reductoisomerase (DXR). |
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Journal, issue, pages | Acs Infect Dis., Vol. 10, Page 1739-1752, Year 2024 |
Publish date | Jun 6, 2023 (structure data deposition date) |
Authors | Abdullaziz, M.A. / Takada, S. / Illarionov, B. / Pessanha de Carvalho, L. / Sakamoto, Y. / Hofmann, S. / Knak, T. / Kiffe-Delf, A.L. / Mazzone, F. / Pfeffer, K. ...Abdullaziz, M.A. / Takada, S. / Illarionov, B. / Pessanha de Carvalho, L. / Sakamoto, Y. / Hofmann, S. / Knak, T. / Kiffe-Delf, A.L. / Mazzone, F. / Pfeffer, K. / Kalscheuer, R. / Bacher, A. / Held, J. / Fischer, M. / Tanaka, N. / Kurz, T. |
External links | Acs Infect Dis. / PubMed:38647213 |
Methods | X-ray diffraction |
Resolution | 1.44 - 1.6 Å |
Structure data | PDB-8jnv: PDB-8jnw: |
Chemicals | ChemComp-MN:
ChemComp-UW0: ChemComp-CA: ChemComp-HOH: ChemComp-NDP: |
Source |
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Keywords | ISOMERASE / Inhibitor / Complex |