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-Structure paper
Title | A bromodomain-independent mechanism of gene regulation by the BET inhibitor JQ1: direct activation of nuclear receptor PXR. |
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Journal, issue, pages | Nucleic Acids Res., Vol. 52, Page 1661-1676, Year 2024 |
Publish date | Nov 15, 2022 (structure data deposition date) |
Authors | Huber, A.D. / Poudel, S. / Wu, J. / Miller, D.J. / Lin, W. / Yang, L. / Bwayi, M.N. / Rimmer, M.A. / Gee, R.R.F. / Seetharaman, J. ...Huber, A.D. / Poudel, S. / Wu, J. / Miller, D.J. / Lin, W. / Yang, L. / Bwayi, M.N. / Rimmer, M.A. / Gee, R.R.F. / Seetharaman, J. / Chai, S.C. / Chen, T. |
External links | Nucleic Acids Res. / PubMed:38084912 |
Methods | X-ray diffraction |
Resolution | 2.15 Å |
Structure data | PDB-8f5y: |
Chemicals | ChemComp-JQ1: ChemComp-HOH: |
Source |
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Keywords | TRANSCRIPTION / nuclear receptor / transcription factor / metabolism / antibiotic |