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-Structure paper
Title | Biochemical and structural basis for the pharmacological inhibition of nuclear hormone receptor PPAR gamma by inverse agonists. |
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Journal, issue, pages | J. Biol. Chem., Vol. 298, Page 102539-102539, Year 2022 |
Publish date | Jul 5, 2022 (structure data deposition date) |
![]() | Irwin, S. / Karr, C. / Furman, C. / Tsai, J. / Gee, P. / Banka, D. / Wibowo, A.S. / Dementiev, A.A. / O'Shea, M. / Yang, J. ...Irwin, S. / Karr, C. / Furman, C. / Tsai, J. / Gee, P. / Banka, D. / Wibowo, A.S. / Dementiev, A.A. / O'Shea, M. / Yang, J. / Lowe, J. / Mitchell, L. / Ruppel, S. / Fekkes, P. / Zhu, P. / Korpal, M. / Larsen, N.A. |
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Methods | X-ray diffraction |
Resolution | 1.59 - 2.95 Å |
Structure data | ![]() PDB-8dkn: ![]() PDB-8dkv: ![]() PDB-8dsy: ![]() PDB-8dsz: |
Chemicals | ![]() ChemComp-EEY: ![]() ChemComp-CXS: ![]() ChemComp-SO4: ![]() ChemComp-HOH: ![]() ChemComp-SKL: ![]() ChemComp-TJC: ![]() ChemComp-TJO: |
Source |
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![]() | NUCLEAR PROTEIN / PPARg / inverse agonist / covalent / T007 / JTP-426467 / H3B-343 / partial agonist / H3B-487 |