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-Structure paper
Title | Discovery of a Potent and Selective CDKL5/GSK3 Chemical Probe That Is Neuroprotective. |
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Journal, issue, pages | Acs Chem Neurosci, Vol. 14, Page 1672-1685, Year 2023 |
Publish date | Feb 9, 2023 (structure data deposition date) |
Authors | Ong, H.W. / Liang, Y. / Richardson, W. / Lowry, E.R. / Wells, C.I. / Chen, X. / Silvestre, M. / Dempster, K. / Silvaroli, J.A. / Smith, J.L. ...Ong, H.W. / Liang, Y. / Richardson, W. / Lowry, E.R. / Wells, C.I. / Chen, X. / Silvestre, M. / Dempster, K. / Silvaroli, J.A. / Smith, J.L. / Wichterle, H. / Pabla, N.S. / Ultanir, S.K. / Bullock, A.N. / Drewry, D.H. / Axtman, A.D. |
External links | Acs Chem Neurosci / PubMed:37084253 |
Methods | X-ray diffraction |
Resolution | 2.2 Å |
Structure data | PDB-8cie: |
Chemicals | ChemComp-US0: ChemComp-SO4: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / KINASE |