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-Structure paper
Title | Modulation of IL-17 backbone dynamics reduces receptor affinity and reveals a new inhibitory mechanism. |
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Journal, issue, pages | Chem Sci, Vol. 14, Page 7524-7536, Year 2023 |
Publish date | Jan 30, 2023 (structure data deposition date) |
![]() | Shaw, D.J. / Waters, L.C. / Strong, S.L. / Schulze, M.E.D. / Greetham, G.M. / Towrie, M. / Parker, A.W. / Prosser, C.E. / Henry, A.J. / Lawson, A.D.G. ...Shaw, D.J. / Waters, L.C. / Strong, S.L. / Schulze, M.E.D. / Greetham, G.M. / Towrie, M. / Parker, A.W. / Prosser, C.E. / Henry, A.J. / Lawson, A.D.G. / Carr, M.D. / Taylor, R.J. / Hunt, N.T. / Muskett, F.W. |
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Methods | X-ray diffraction |
Resolution | 2.9 Å |
Structure data | ![]() PDB-8cdg: |
Chemicals | ![]() ChemComp-UTF: |
Source |
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![]() | CYTOKINE / inhibitor / complex / macrocycle |