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-Structure paper
Title | Discovery of a Potent and Selective Naphthyridine-Based Chemical Probe for Casein Kinase 2. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 14, Page 432-441, Year 2023 |
Publish date | Oct 27, 2022 (structure data deposition date) |
Authors | Davis-Gilbert, Z.W. / Kramer, A. / Dunford, J.E. / Howell, S. / Senbabaoglu, F. / Wells, C.I. / Bashore, F.M. / Havener, T.M. / Smith, J.L. / Hossain, M.A. ...Davis-Gilbert, Z.W. / Kramer, A. / Dunford, J.E. / Howell, S. / Senbabaoglu, F. / Wells, C.I. / Bashore, F.M. / Havener, T.M. / Smith, J.L. / Hossain, M.A. / Oppermann, U. / Drewry, D.H. / Axtman, A.D. |
External links | Acs Med. Chem. Lett. / PubMed:37077385 |
Methods | X-ray diffraction |
Resolution | 2.8 Å |
Structure data | PDB-8bgc: |
Chemicals | ChemComp-SO4: ChemComp-QIA: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / CK2apha / Kinase |