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-Structure paper
Title | Insights on JAK2 Modulation by Potent, Selective, and Cell-Permeable Pseudokinase-Domain Ligands. |
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Journal, issue, pages | J. Med. Chem., Vol. 65, Page 8380-8400, Year 2022 |
Publish date | Nov 30, 2021 (structure data deposition date) |
Authors | Liosi, M.E. / Ippolito, J.A. / Henry, S.P. / Krimmer, S.G. / Newton, A.S. / Cutrona, K.J. / Olivarez, R.A. / Mohanty, J. / Schlessinger, J. / Jorgensen, W.L. |
External links | J. Med. Chem. / PubMed:35653642 |
Methods | X-ray diffraction |
Resolution | 2.04 Å |
Structure data | PDB-7t0p: |
Chemicals | ChemComp-E3W: ChemComp-GOL: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE/INHIBITOR / PSEUDOKINASE DOMAIN / INHIBITOR / COMPLEX / TRANSFERASE / TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX / SIGNALING PROTEIN / TRANSFERASE-INHIBITOR complex |