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-Structure paper
Title | Filling a nick in NIK: Extending the half-life of a NIK inhibitor through structure-based drug design. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 89, Page 129277-129277, Year 2023 |
Publish date | Nov 29, 2021 (structure data deposition date) |
Authors | Crawford, J.J. / Feng, J. / Brightbill, H.D. / Johnson, A.R. / Wright, M. / Kolesnikov, A. / Lee, W. / Castanedo, G.M. / Do, S. / Blaquiere, N. ...Crawford, J.J. / Feng, J. / Brightbill, H.D. / Johnson, A.R. / Wright, M. / Kolesnikov, A. / Lee, W. / Castanedo, G.M. / Do, S. / Blaquiere, N. / Staben, S.T. / Chiang, P.C. / Fan, P.W. / Baumgardner, M. / Wong, S. / Godemann, R. / Grabbe, A. / Wiegel, C. / Sujatha-Bhaskar, S. / Hymowitz, S.G. / Liau, N. / Hsu, P.L. / McEwan, P.A. / Ismaili, M.H.A. / Landry, M.L. |
External links | Bioorg. Med. Chem. Lett. / PubMed:37105490 |
Methods | X-ray diffraction |
Resolution | 2.8 Å |
Structure data | PDB-7szr: |
Chemicals | ChemComp-SO4: ChemComp-DYQ: |
Source |
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Keywords | SIGNALING PROTEIN / Kinase / inhibitor / NF-kB inducing kinase |