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-Structure paper
Title | Structure-Guided Development of Small-Molecule PRC2 Inhibitors Targeting EZH2-EED Interaction. |
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Journal, issue, pages | J. Med. Chem., Vol. 64, Page 8194-8207, Year 2021 |
Publish date | Dec 4, 2020 (structure data deposition date) |
![]() | Du, D. / Xu, D. / Zhu, L. / Stazi, G. / Zwergel, C. / Liu, Y. / Luo, Z. / Li, Y. / Zhang, Y. / Zhu, K. ...Du, D. / Xu, D. / Zhu, L. / Stazi, G. / Zwergel, C. / Liu, Y. / Luo, Z. / Li, Y. / Zhang, Y. / Zhu, K. / Ding, Y. / Liu, J. / Fan, S. / Zhao, K. / Zhang, N. / Kong, X. / Jiang, H. / Chen, K. / Valente, S. / Min, J. / Duan, W. / Luo, C. |
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Methods | X-ray diffraction |
Resolution | 2.15 Å |
Structure data | ![]() PDB-7kxt: |
Chemicals | ![]() ChemComp-XB7: ![]() ChemComp-UNX: ![]() ChemComp-HOH: |
Source |
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![]() | GENE REGULATION / EED / WD40 / Structural Genomics / Structural Genomics Consortium / SGC |