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-Structure paper
Title | A selective WDR5 degrader inhibits acute myeloid leukemia in patient-derived mouse models. |
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Journal, issue, pages | Sci Transl Med, Vol. 13, Page eabj1578-eabj1578, Year 2021 |
Publish date | Aug 18, 2020 (structure data deposition date) |
![]() | Yu, X. / Li, D. / Kottur, J. / Shen, Y. / Kim, H.S. / Park, K.S. / Tsai, Y.H. / Gong, W. / Wang, J. / Suzuki, K. ...Yu, X. / Li, D. / Kottur, J. / Shen, Y. / Kim, H.S. / Park, K.S. / Tsai, Y.H. / Gong, W. / Wang, J. / Suzuki, K. / Parker, J. / Herring, L. / Kaniskan, H.U. / Cai, L. / Jain, R. / Liu, J. / Aggarwal, A.K. / Wang, G.G. / Jin, J. |
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Methods | X-ray diffraction |
Resolution | 1.7 - 2.12 Å |
Structure data | ![]() PDB-7jto: ![]() PDB-7jtp: |
Chemicals | ![]() ChemComp-SCN: ![]() ChemComp-EDO: ![]() ChemComp-VKA: ![]() ChemComp-GOL: ![]() ChemComp-NA: ![]() ChemComp-HOH: ![]() ChemComp-X6M: |
Source |
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![]() | PROTEIN BINDING / Protac / protein degradation / ubiquitination |