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Title | Discovery of SARS-CoV-2 Papain-like Protease Inhibitors through a Combination of High-Throughput Screening and a FlipGFP-Based Reporter Assay. |
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Journal, issue, pages | Acs Cent. Sci., Vol. 7, Page 1245-1260, Year 2021 |
Publish date | Aug 12, 2020 (structure data deposition date) |
Authors | Ma, C. / Sacco, M.D. / Xia, Z. / Lambrinidis, G. / Townsend, J.A. / Hu, Y. / Meng, X. / Szeto, T. / Ba, M. / Zhang, X. ...Ma, C. / Sacco, M.D. / Xia, Z. / Lambrinidis, G. / Townsend, J.A. / Hu, Y. / Meng, X. / Szeto, T. / Ba, M. / Zhang, X. / Gongora, M. / Zhang, F. / Marty, M.T. / Xiang, Y. / Kolocouris, A. / Chen, Y. / Wang, J. |
External links | Acs Cent. Sci. / PubMed:34341772 |
Methods | X-ray diffraction |
Resolution | 2.48 Å |
Structure data | PDB-7jrn: |
Chemicals | ChemComp-TTT: ChemComp-ZN: ChemComp-SO4: ChemComp-HOH: |
Source |
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Keywords | VIRAL PROTEIN / COVID / COVID19 / COVID-19 / SARS / SARS COV2 / COV / NCOV 19 / CORONAVIRUS / MAIN PROTEASE / 3CL / MPRO / PRO / GC376 / calpain inhibitor II / leupeptin / calpain / aldehyde / GC-376 / 3cl-like / a-ketoamide / alpheketoamide / alpha / ketoamide / PEPTIDOMIMETIC / PROTEASE / CYSTEINE / HYDROLASE-HYDROLASE INHIBITOR complex / GRL0617 / papin-like protease / PLP / PLPro / PL-pro / papain |