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-Structure paper
Title | Potent and Selective RIPK1 Inhibitors Targeting Dual-Pockets for the Treatment of Systemic Inflammatory Response Syndrome and Sepsis. |
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Journal, issue, pages | Angew. Chem. Int. Ed. Engl., Vol. 61, Page e202114922-e202114922, Year 2022 |
Publish date | Jul 15, 2021 (structure data deposition date) |
![]() | Yang, X. / Lu, H. / Xie, H. / Zhang, B. / Nie, T. / Fan, C. / Yang, T. / Xu, Y. / Su, H. / Tang, W. / Zhou, B. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2 - 2.21 Å |
Structure data | ![]() PDB-7fcz: ![]() PDB-7fd0: |
Chemicals | ![]() ChemComp-3IF: ![]() ChemComp-HOH: ![]() ChemComp-3IU: |
Source |
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![]() | IMMUNE SYSTEM/INHIBITOR / IMMUNE SYSTEM-INHIBITOR COMPLEX |