+Search query
-Structure paper
Title | Structure Base Design of A new chemotype of Four-Cycle Compounds as Bromodomain and Extra-Terminal (BET) Inhibitors with The Second Bromodomain Bias and Highly Anti-inflammatory Potency |
---|---|
Journal, issue, pages | To Be Published |
Publish date | Dec 20, 2020 (structure data deposition date) |
![]() | Li, Z. / Lu, T. / Chen, P. / Luo, C. / Zgou, B. |
![]() | Search PubMed |
Methods | X-ray diffraction |
Resolution | 1.79998842375 - 2.29994028999 Å |
Structure data | ![]() PDB-7dpn: ![]() PDB-7dpo: |
Chemicals | ![]() ChemComp-HFU: ![]() ChemComp-HOH: |
Source |
|
![]() | ANTITUMOR PROTEIN / Antitumor; BET proteins; Bromodomain inhibitor; Epigenetic readers |