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-Structure paper
Title | Discovery of a Novel Class of Covalent Dual Inhibitors Targeting the Protein Kinases BMX and BTK. |
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Journal, issue, pages | Int J Mol Sci, Vol. 21, Year 2020 |
Publish date | Oct 16, 2020 (structure data deposition date) |
Authors | Forster, M. / Liang, X.J. / Schroder, M. / Gerstenecker, S. / Chaikuad, A. / Knapp, S. / Laufer, S. / Gehringer, M. |
External links | Int J Mol Sci / PubMed:33291717 |
Methods | X-ray diffraction |
Resolution | 1.95 - 2.4 Å |
Structure data | PDB-7apf: PDB-7apg: |
Chemicals | ChemComp-RQZ: ChemComp-PHU: ChemComp-EDO: ChemComp-HOH: ChemComp-RQT: |
Source |
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Keywords | TRANSFERASE / kinase / JAK3 / inhibitor / covalent inhibitor / Structural Genomics / Structural Genomics Consortium / SGC |