+Search query
-Structure paper
Title | Pan-SMARCA/PB1 Bromodomain Inhibitors and Their Role in Regulating Adipogenesis. |
---|---|
Journal, issue, pages | J. Med. Chem., Vol. 63, Page 14680-14699, Year 2020 |
Publish date | Jul 6, 2020 (structure data deposition date) |
Authors | Wanior, M. / Preuss, F. / Ni, X. / Kramer, A. / Mathea, S. / Gobel, T. / Heidenreich, D. / Simonyi, S. / Kahnt, A.S. / Joerger, A.C. / Knapp, S. |
External links | J. Med. Chem. / PubMed:33216538 |
Methods | X-ray diffraction |
Resolution | 1.14 - 2.02 Å |
Structure data | PDB-6zn6: PDB-6znv: PDB-6zs2: PDB-6zs3: PDB-6zs4: |
Chemicals | ChemComp-QMT: ChemComp-EDO: ChemComp-HOH: ChemComp-QMW: ChemComp-ZN: ChemComp-CL: ChemComp-ACT: ChemComp-FX5: ChemComp-QP8: |
Source |
|
Keywords | PROTEIN BINDING / Bromodomain Inhibitor Epigenetics / GENE REGULATION / BROMODOMAIN / ATP-DEPENDENT HELICASE SMARCA4 / BRG1-ASSOCIATED FACTOR 190A / BAF190A / MITOTIC GROWTH AND TRANSCRIPTION ACTIVATOR / PROTEIN BRG-1 / PROTEIN BRAHMA HOMOLOG 1 / SNF2-BETA / SWI/SNF-RELATED MATRIX-ASSOCIATED ACTIN-DEPENDENT REGULATOR OF CHROMATIN SUBFAMILY A MEMBER 4 / STRUCTURAL GENOMICS CONSORTIUM / SGC / TRANSCRIPTION / COMPLEX / SMALL MOLECULE |