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-Structure paper
Title | Computationally designed peptide macrocycle inhibitors of New Delhi metallo-beta-lactamase 1. |
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Journal, issue, pages | Proc. Natl. Acad. Sci. USA, Vol. 118, Year 2021 |
Publish date | Jun 5, 2020 (structure data deposition date) |
![]() | Mulligan, V.K. / Workman, S. / Sun, T. / Rettie, S. / Li, X. / Worrall, L.J. / Craven, T.W. / King, D.T. / Hosseinzadeh, P. / Watkins, A.M. ...Mulligan, V.K. / Workman, S. / Sun, T. / Rettie, S. / Li, X. / Worrall, L.J. / Craven, T.W. / King, D.T. / Hosseinzadeh, P. / Watkins, A.M. / Renfrew, P.D. / Guffy, S. / Labonte, J.W. / Moretti, R. / Bonneau, R. / Strynadka, N.C.J. / Baker, D. |
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Methods | X-ray diffraction |
Resolution | 1.6 - 2.2 Å |
Structure data | ![]() PDB-6xbe: ![]() PDB-6xbf: ![]() PDB-6xci: |
Chemicals | ![]() ChemComp-ZN: ![]() ChemComp-HOH: ![]() ChemComp-ACT: ![]() ChemComp-CD: |
Source |
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![]() | HYDROLASE/HYDROLASE INHIBITOR / Cyclic peptide / macrocycle inhibitor / ANTIBIOTIC / HYDROLASE-HYDROLASE INHIBITOR complex |