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-Structure paper
Title | Discovery ofN-(Indazol-3-yl)piperidine-4-carboxylic Acids as ROR gamma t Allosteric Inhibitors for Autoimmune Diseases. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 11, Page 114-119, Year 2020 |
Publish date | Sep 16, 2019 (structure data deposition date) |
Authors | Zhang, H. / Lapointe, B.T. / Anthony, N. / Azevedo, R. / Cals, J. / Correll, C.C. / Daniels, M. / Deshmukh, S. / van Eenenaam, H. / Ferguson, H. ...Zhang, H. / Lapointe, B.T. / Anthony, N. / Azevedo, R. / Cals, J. / Correll, C.C. / Daniels, M. / Deshmukh, S. / van Eenenaam, H. / Ferguson, H. / Hegde, L.G. / Karstens, W.J. / Maclean, J. / Miller, J.R. / Moy, L.Y. / Simov, V. / Nagpal, S. / Oubrie, A. / Palte, R.L. / Parthasarathy, G. / Sciammetta, N. / van der Stelt, M. / Woodhouse, J.D. / Trotter, B.W. / Barr, K. |
External links | Acs Med. Chem. Lett. / PubMed:32071676 |
Methods | X-ray diffraction |
Resolution | 2.87 Å |
Structure data | PDB-6ucg: |
Chemicals | ChemComp-Q3Y: ChemComp-HOH: |
Source |
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Keywords | TRANSCRIPTION / ROR gamma T / allosteric / nuclear receptor |