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-Structure paper
Title | Identification and Optimization of EphA2-Selective Bicycles for the Delivery of Cytotoxic Payloads. |
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Journal, issue, pages | J. Med. Chem., Vol. 63, Page 4107-4116, Year 2020 |
Publish date | Jun 3, 2019 (structure data deposition date) |
Authors | Mudd, G.E. / Brown, A. / Chen, L. / van Rietschoten, K. / Watcham, S. / Teufel, D.P. / Pavan, S. / Lani, R. / Huxley, P. / Bennett, G.S. |
External links | J. Med. Chem. / PubMed:32202781 |
Methods | X-ray diffraction |
Resolution | 2.26 Å |
Structure data | PDB-6rw2: |
Chemicals | ChemComp-GOL: ChemComp-29N: ChemComp-HOH: |
Source |
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Keywords | SIGNALING PROTEIN / EphA2 / inhibitor / complex |