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-Structure paper
Title | Identification of a RIP1 Kinase Inhibitor Clinical Candidate (GSK3145095) for the Treatment of Pancreatic Cancer. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 10, Page 857-862, Year 2019 |
Publish date | May 2, 2019 (structure data deposition date) |
![]() | Harris, P.A. / Marinis, J.M. / Lich, J.D. / Berger, S.B. / Chirala, A. / Cox, J.A. / Eidam, P.M. / Finger, J.N. / Gough, P.J. / Jeong, J.U. ...Harris, P.A. / Marinis, J.M. / Lich, J.D. / Berger, S.B. / Chirala, A. / Cox, J.A. / Eidam, P.M. / Finger, J.N. / Gough, P.J. / Jeong, J.U. / Kang, J. / Kasparcova, V. / Leister, L.K. / Mahajan, M.K. / Miller, G. / Nagilla, R. / Ouellette, M.T. / Reilly, M.A. / Rendina, A.R. / Rivera, E.J. / Sun, H.H. / Thorpe, J.H. / Totoritis, R.D. / Wang, W. / Wu, D. / Zhang, D. / Bertin, J. / Marquis, R.W. |
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Methods | X-ray diffraction |
Resolution | 2.87 Å |
Structure data | ![]() PDB-6rln: |
Chemicals | ![]() ChemComp-K8K: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE / Inhibitor / Complex |