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-Structure paper
Title | Discovery of 2-phenoxyacetamides as inhibitors of the Wnt-depalmitoleating enzyme NOTUM from an X-ray fragment screen. |
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Journal, issue, pages | Medchemcomm, Vol. 10, Page 1361-1369, Year 2019 |
Publish date | Apr 2, 2019 (structure data deposition date) |
![]() | Atkinson, B.N. / Steadman, D. / Zhao, Y. / Sipthorp, J. / Vecchia, L. / Ruza, R.R. / Jeganathan, F. / Lines, G. / Frew, S. / Monaghan, A. ...Atkinson, B.N. / Steadman, D. / Zhao, Y. / Sipthorp, J. / Vecchia, L. / Ruza, R.R. / Jeganathan, F. / Lines, G. / Frew, S. / Monaghan, A. / Kjær, S. / Bictash, M. / Jones, E.Y. / Fish, P.V. |
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Methods | X-ray diffraction |
Resolution | 1.27 - 1.5 Å |
Structure data | ![]() PDB-6r8p: ![]() PDB-6r8q: ![]() PDB-6r8r: |
Chemicals | ![]() ChemComp-NAG: ![]() ChemComp-GOL: ![]() ChemComp-SO4: ![]() ChemComp-DMS: ![]() ChemComp-JVB: ![]() ChemComp-HOH: ![]() ChemComp-EDO: ![]() ChemComp-JV5: ![]() ChemComp-JV8: |
Source |
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![]() | HYDROLASE / Notum inhibitor / Wnt signalling / Crystallographic Fragment Screen |