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-Structure paper
Title | Engineered Carbonic Anhydrase VI-Mimic Enzyme Switched the Structure and Affinities of Inhibitors. |
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Journal, issue, pages | Sci Rep, Vol. 9, Page 12710-12710, Year 2019 |
Publish date | Jan 31, 2019 (structure data deposition date) |
Authors | Kazokaite, J. / Kairys, V. / Smirnoviene, J. / Smirnov, A. / Manakova, E. / Tolvanen, M. / Parkkila, S. / Matulis, D. |
External links | Sci Rep / PubMed:31481705 |
Methods | X-ray diffraction |
Resolution | 1.3 - 1.42 Å |
Structure data | PDB-6ql1: PDB-6ql2: PDB-6ql3: |
Chemicals | ChemComp-ZN: ChemComp-DMS: ChemComp-EDO: ChemComp-BCN: ChemComp-V50: ChemComp-NA: ChemComp-HOH: ChemComp-MES: ChemComp-EZL: ChemComp-V14: ChemComp-PEG: ChemComp-MLA: ChemComp-BEZ: |
Source |
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Keywords | LYASE / drug design / carbonic anhydrase / benzenesulfonamide / metal-binding / lyase-lyase inhibitor complex |