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-Structure paper
Title | Dual Inhibition of TAF1 and BET Bromodomains from the BI-2536 Kinase Inhibitor Scaffold. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 10, Page 1443-1449, Year 2019 |
Publish date | May 23, 2019 (structure data deposition date) |
Authors | Remillard, D. / Buckley, D.L. / Seo, H.S. / Ferguson, F.M. / Dhe-Paganon, S. / Bradner, J.E. / Gray, N.S. |
External links | Acs Med. Chem. Lett. / PubMed:31620231 |
Methods | X-ray diffraction |
Resolution | 2.8 Å |
Structure data | PDB-6p38: |
Chemicals | ChemComp-NQV: |
Source |
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Keywords | TRANSFERASE / kinase / bromodomain / inhibitor / TRANSCRIPTION |