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Title | The Selective Tie2 Inhibitor Rebastinib Blocks Recruitment and Function of Tie2 |
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Journal, issue, pages | Mol. Cancer Ther., Vol. 16, Page 2486-2501, Year 2017 |
Publish date | Oct 29, 2018 (structure data deposition date) |
Authors | Harney, A.S. / Karagiannis, G.S. / Pignatelli, J. / Smith, B.D. / Kadioglu, E. / Wise, S.C. / Hood, M.M. / Kaufman, M.D. / Leary, C.B. / Lu, W.P. ...Harney, A.S. / Karagiannis, G.S. / Pignatelli, J. / Smith, B.D. / Kadioglu, E. / Wise, S.C. / Hood, M.M. / Kaufman, M.D. / Leary, C.B. / Lu, W.P. / Al-Ani, G. / Chen, X. / Entenberg, D. / Oktay, M.H. / Wang, Y. / Chun, L. / De Palma, M. / Jones, J.G. / Flynn, D.L. / Condeelis, J.S. |
External links | Mol. Cancer Ther. / PubMed:28838996 |
Methods | X-ray diffraction |
Resolution | 2.05 Å |
Structure data | PDB-6mwe: |
Chemicals | ChemComp-SO4: ChemComp-919: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / TIE2 / DP1919 / EMERALDBIO / DECIPHERA |