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Title | Fragment-based Discovery of a Small-Molecule Protein Kinase C-iota Inhibitor Binding Post-kinase Domain Residues. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 10, Page 318-323, Year 2019 |
Publish date | Oct 21, 2018 (structure data deposition date) |
Authors | Kwiatkowski, J. / Baburajendran, N. / Poulsen, A. / Liu, B. / Tee, D.H.Y. / Wong, Y.X. / Poh, Z.Y. / Ong, E.H. / Dinie, N. / Cherian, J. ...Kwiatkowski, J. / Baburajendran, N. / Poulsen, A. / Liu, B. / Tee, D.H.Y. / Wong, Y.X. / Poh, Z.Y. / Ong, E.H. / Dinie, N. / Cherian, J. / Jansson, A.E. / Hill, J. / Keller, T.H. / Hung, A.W. |
External links | Acs Med. Chem. Lett. / PubMed:30891133 |
Methods | X-ray diffraction |
Resolution | 3.261 Å |
Structure data | PDB-6ilz: |
Chemicals | ChemComp-AFU: |
Source |
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Keywords | TRANSFERASE / Kinase / Atypical kinase / phosphorylation / inhibitor / PKCiota / iota type / kinase domain |