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-Structure paper
Title | Activation loop targeting strategy for design of receptor-interacting protein kinase 2 (RIPK2) inhibitors. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 28, Page 577-583, Year 2018 |
Publish date | Oct 19, 2017 (structure data deposition date) |
Authors | Suebsuwong, C. / Pinkas, D.M. / Ray, S.S. / Bufton, J.C. / Dai, B. / Bullock, A.N. / Degterev, A. / Cuny, G.D. |
External links | Bioorg. Med. Chem. Lett. / PubMed:29409752 |
Methods | X-ray diffraction |
Resolution | 2.38 Å |
Structure data | PDB-6es0: |
Chemicals | ChemComp-BW8: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / Kinase Inhibitor |