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-Structure paper
Title | Design and Evaluation of Highly Selective Human Immunoproteasome Inhibitors Reveal a Compensatory Process That Preserves Immune Cell Viability. |
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Journal, issue, pages | J. Med. Chem., Vol. 62, Page 7032-7041, Year 2019 |
Publish date | Jul 19, 2018 (structure data deposition date) |
![]() | Ladi, E. / Everett, C. / Stivala, C.E. / Daniels, B.E. / Durk, M.R. / Harris, S.F. / Huestis, M.P. / Purkey, H.E. / Staben, S.T. / Augustin, M. ...Ladi, E. / Everett, C. / Stivala, C.E. / Daniels, B.E. / Durk, M.R. / Harris, S.F. / Huestis, M.P. / Purkey, H.E. / Staben, S.T. / Augustin, M. / Blaesse, M. / Steinbacher, S. / Eidenschenk, C. / Pappu, R. / Siu, M. |
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Methods | X-ray diffraction |
Resolution | 2.77 Å |
Structure data | ![]() PDB-6e5b: |
Chemicals | ![]() ChemComp-SCN: ![]() ChemComp-NA: ![]() ChemComp-HUJ: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE / MULTICATALYTIC PROTEINASE / 20S PROTEASOME / PROTEASE / PROTEROS / PROTEROS BIOSTRUCTURES GMBH |