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-Structure paper
Title | Single and Dual Targeting of Mutant EGFR with an Allosteric Inhibitor. |
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Journal, issue, pages | Cancer Discov, Vol. 9, Page 926-943, Year 2019 |
Publish date | Jun 21, 2018 (structure data deposition date) |
![]() | To, C. / Jang, J. / Chen, T. / Park, E. / Mushajiang, M. / De Clercq, D.J.H. / Xu, M. / Wang, S. / Cameron, M.D. / Heppner, D.E. ...To, C. / Jang, J. / Chen, T. / Park, E. / Mushajiang, M. / De Clercq, D.J.H. / Xu, M. / Wang, S. / Cameron, M.D. / Heppner, D.E. / Shin, B.H. / Gero, T.W. / Yang, A. / Dahlberg, S.E. / Wong, K.K. / Eck, M.J. / Gray, N.S. / Janne, P.A. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.2 Å |
Structure data | ![]() PDB-6duk: |
Chemicals | ![]() ChemComp-MG: ![]() ChemComp-ANP: ![]() ChemComp-JBJ: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / Allosteric inhibitor / EGFR / ONCOPROTEIN / TRANSFERASE-TRANSFERASE INHIBITOR complex |