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Title | Structure-Guided Design and Procognitive Assessment of a Potent and Selective Phosphodiesterase 2A Inhibitor. |
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Journal, issue, pages | ACS Med Chem Lett, Vol. 9, Page 815-820, Year 2018 |
Publish date | Apr 5, 2018 (structure data deposition date) |
Authors | Stachel, S.J. / Berger, R. / Nomland, A.B. / Ginnetti, A.T. / Paone, D.V. / Wang, D. / Puri, V. / Lange, H. / Drott, J. / Lu, J. ...Stachel, S.J. / Berger, R. / Nomland, A.B. / Ginnetti, A.T. / Paone, D.V. / Wang, D. / Puri, V. / Lange, H. / Drott, J. / Lu, J. / Marcus, J. / Dwyer, M.P. / Suon, S. / Uslaner, J.M. / Smith, S.M. |
External links | ACS Med Chem Lett / PubMed:30128073 |
Methods | X-ray diffraction |
Resolution | 1.54 - 1.69 Å |
Structure data | PDB-6cyb: PDB-6cyc: PDB-6cyd: |
Chemicals | ChemComp-ZN: ChemComp-MG: ChemComp-EDO: ChemComp-FKV: ChemComp-HOH: ChemComp-FKJ: ChemComp-FKG: |
Source |
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Keywords | HYDROLASE/HYDROLASE INHIBITOR / PDE2 / inhibition / structure-guided design / HYDROLASE-HYDROLASE INHIBITOR complex |