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-Structure paper
Title | Identification of Potent and Selective RIPK2 Inhibitors for the Treatment of Inflammatory Diseases. |
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Journal, issue, pages | ACS Med Chem Lett, Vol. 8, Page 1048-1053, Year 2017 |
Publish date | Jun 15, 2017 (structure data deposition date) |
Authors | He, X. / Da Ros, S. / Nelson, J. / Zhu, X. / Jiang, T. / Okram, B. / Jiang, S. / Michellys, P.Y. / Iskandar, M. / Espinola, S. ...He, X. / Da Ros, S. / Nelson, J. / Zhu, X. / Jiang, T. / Okram, B. / Jiang, S. / Michellys, P.Y. / Iskandar, M. / Espinola, S. / Jia, Y. / Bursulaya, B. / Kreusch, A. / Gao, M.Y. / Spraggon, G. / Baaten, J. / Clemmer, L. / Meeusen, S. / Huang, D. / Hill, R. / Nguyen-Tran, V. / Fathman, J. / Liu, B. / Tuntland, T. / Gordon, P. / Hollenbeck, T. / Ng, K. / Shi, J. / Bordone, L. / Liu, H. |
External links | ACS Med Chem Lett / PubMed:29057049 |
Methods | X-ray diffraction |
Resolution | 2.85 - 2.89 Å |
Structure data | PDB-5w5j: PDB-5w5o: |
Chemicals | ChemComp-9WS: ChemComp-SO4: ChemComp-HOH: ChemComp-9XA: |
Source |
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Keywords | HYDROLASE/HYDROLASE INHIBITOR / Inhibitor / Complex / Kinase / HYDROLASE / HYDROLASE-HYDROLASE INHIBITOR complex / Transferase/Transferase Inhibitor / Tetartohedral winning / Transferase-Transferase Inhibitor complex |