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-Structure paper
Title | Metallacarborane Sulfamides: Unconventional, Specific, and Highly Selective Inhibitors of Carbonic Anhydrase IX. |
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Journal, issue, pages | J. Med. Chem., Year 2019 |
Publish date | Jul 13, 2017 (structure data deposition date) |
Authors | Gruner, B. / Brynda, J. / Das, V. / Sicha, V. / Stepankova, J. / Nekvinda, J. / Holub, J. / Pospisilova, K. / Fabry, M. / Pachl, P. ...Gruner, B. / Brynda, J. / Das, V. / Sicha, V. / Stepankova, J. / Nekvinda, J. / Holub, J. / Pospisilova, K. / Fabry, M. / Pachl, P. / Kral, V. / Kugler, M. / Masek, V. / Medvedikova, M. / Matejkova, S. / Nova, A. / Liskova, B. / Gurska, S. / Dzubak, P. / Hajduch, M. / Rezacova, P. |
External links | J. Med. Chem. / PubMed:31568723 |
Methods | X-ray diffraction |
Resolution | 1.1 Å |
Structure data | PDB-5ogn: PDB-5ogp: |
Chemicals | ChemComp-ZN: ChemComp-B8B: ChemComp-HOH: ChemComp-9UK: |
Source |
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Keywords | LYASE / Carbonic Anhydrase IX / CA Inhibitor |