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-Structure paper
Title | Direct NMR Probing of Hydration Shells of Protein Ligand Interfaces and Its Application to Drug Design. |
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Journal, issue, pages | J. Med. Chem., Vol. 60, Page 8708-8715, Year 2017 |
Publish date | Oct 14, 2016 (structure data deposition date) |
Authors | Geist, L. / Mayer, M. / Cockcroft, X.L. / Wolkerstorfer, B. / Kessler, D. / Engelhardt, H. / McConnell, D.B. / Konrat, R. |
External links | J. Med. Chem. / PubMed:28910100 |
Methods | X-ray diffraction |
Resolution | 1.38 - 1.65 Å |
Structure data | PDB-5m39: PDB-5m3a: |
Chemicals | ChemComp-7EA: ChemComp-HOH: ChemComp-EDO: ChemComp-7E7: |
Source |
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Keywords | TRANSCRIPTION / BROMODOMAIN / BRD4 BD1 / EPIGENETIC / HISTONE READER |