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Title | SETDB1 in complex with an early stage, low affinity fragment candidate modelled at reduced occupancy |
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Journal, issue, pages | To Be Published |
Publish date | Jun 6, 2016 (structure data deposition date) |
![]() | Tempel, W. / Harding, R.J. / Mader, P. / Dobrovetsky, E. / Walker, J.R. / Brown, P.J. / Schapira, M. / Arrowsmith, C.H. / Edwards, A.M. / Santhakumar, S. / Structural Genomics Consortium (SGC) |
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Methods | X-ray diffraction |
Resolution | 1.47 - 1.7 Å |
Structure data | ![]() PDB-5kch: ![]() PDB-5kco: |
Chemicals | ![]() ChemComp-UNX: ![]() ChemComp-DMS: ![]() ChemComp-SO4: ![]() ChemComp-6RN: ![]() ChemComp-HOH: ![]() ChemComp-6RO: |
Source |
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![]() | TRANSFERASE / Fragment Screening / DIAMOND I04-1 XCHEM / PANDDA / Structural Genomics / Structural Genomics Consortium / SGC |