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-Structure paper
Title | Design and characterization of bivalent BET inhibitors. |
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Journal, issue, pages | Nat. Chem. Biol., Vol. 12, Page 1089-1096, Year 2016 |
Publish date | May 12, 2016 (structure data deposition date) |
Authors | Tanaka, M. / Roberts, J.M. / Seo, H.S. / Souza, A. / Paulk, J. / Scott, T.G. / DeAngelo, S.L. / Dhe-Paganon, S. / Bradner, J.E. |
External links | Nat. Chem. Biol. / PubMed:27775715 |
Methods | X-ray diffraction |
Resolution | 1.71 Å |
Structure data | PDB-5jwm: |
Chemicals | ChemComp-6ON: ChemComp-HOH: |
Source |
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Keywords | transcription/transcription inhibitor / bivalent-ligand / bromodomain / inhibitor / transcription-transcription inhibitor complex |